Khoom Taw Qhia:
TBB (CAS: 17374-26-}4) yog ib tug classic cell-permeable, ATP-kev sib tw xaiv inhibitor ntawm casein kinase 2 (Casein Kinase 2, CK2/CK2 ), thiab yog siv nyob rau hauv kev tshawb fawb.
Daim ntawv thov:
1. Nws tuaj yeem siv rau kev kawm ntawm CK2 signaling pathway, los tshawb txog kev tswj lub voj voog ntawm tes, kho DNA puas, Wnt/ -catenin signaling thiab transcriptional regulation nrog CK2.
2. Nws tuaj yeem siv los ua kev tswj xyuas kev tshuaj ntsuam kinase, ua haujlwm raws li CK2-kev sojntsuam tshwj xeeb, rau kev kuaj xyuas tshwj xeeb ntawm 33 hom Ser / Thr thiab Tyr protein kinases.
3. Nws tuaj yeem siv rau hauv cell - kev sim qib thiab kev sim tsiaj qauv.
Ntim:
Ntim raws li tus neeg siv khoom xav tau.
Cia tej yam kev mob:
Khaws kaw, khaws cia ntawm -20 degree, kom qhuav thiab deb ntawm lub teeb, nyob rau hauv kev tiv thaiv roj inert.
Chaw thau khoom thiab thauj khoom:
Hiav txwv los yog Cua
Qhov zoo:
1. High chemical stability thiab thermal stability;
2. Kev cai Synthesis;
3. Kev tswj xyuas nruj thiab kev txhawb nqa kev ua raws cai;
4. Kev teb sai thiab kev txhawb nqa.
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